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Academic Journal

Aryl amino acetamides prevent Plasmodium falciparum ring development via targeting the lipid-transfer protein PfSTART1.

  • Authors : Dans MG; Burnet Institute, Melbourne, VIC, 3004, Australia. .; Walter and Eliza Hall Institute, Parkville, VIC, 3052, Australia. .

Subjects: Plasmodium falciparum*/Plasmodium falciparum*/Plasmodium falciparum*/drug effects ; Plasmodium falciparum*/Plasmodium falciparum*/Plasmodium falciparum*/genetics ; Plasmodium falciparum*/Plasmodium falciparum*/Plasmodium falciparum*/metabolism

  • Source: Nature communications [Nat Commun] 2024 Jun 18; Vol. 15 (1), pp. 5219. Date of Electronic Publication: 2024 Jun 18.Publisher: Nature Pub. Group Country of Publication: England NLM ID: 101528555 Publication Model: Electronic Cited Medium: Internet ISSN:

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Academic Journal

Design and Synthesis of 2-Phenylindolizine Acetamides: Molecular Docking, in Vitro Antimicrobial and Anticancer Activity Evaluation.

  • Authors : Kumar Gandham S; Department of Chemistry, GITAM School of Science, GITAM (Deemed to be University), Gandhi Nagar, Rushikonda, Visakhapatnam, Andhra Pradesh-530045, India.; Jha A

Subjects: Acetamides*/Acetamides*/Acetamides*/chemistry ; Acetamides*/Acetamides*/Acetamides*/pharmacology ; Acetamides*/Acetamides*/Acetamides*/chemical synthesis

  • Source: Chemistry & biodiversity [Chem Biodivers] 2024 May; Vol. 21 (5), pp. e202400075. Date of Electronic Publication: 2024 Mar 28.Publisher: Verlag Helvetica Chimica Acta Country of Publication: Switzerland NLM ID: 101197449 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Design, Synthesis, and Structure-Activity Relationship Studies of Novel GPR88 Agonists (4-Substituted-phenyl)acetamides Based on the Reversed Amide Scaffold.

  • Authors : Rahman MT; Center for Drug Discovery, Research Triangle Institute, Research Triangle Park, North Carolina 27709, United States.; Guan D

Subjects: Acetamides*/Acetamides*/Acetamides*/pharmacology ; Amides* ; Receptors, G-Protein-Coupled*/Receptors, G-Protein-Coupled*/Receptors, G-Protein-Coupled*/agonists

  • Source: ACS chemical neuroscience [ACS Chem Neurosci] 2024 Jan 03; Vol. 15 (1), pp. 169-192. Date of Electronic Publication: 2023 Dec 12.Publisher: American Chemical Society Country of Publication: United States NLM ID: 101525337 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

2-(Methyl(phenyl)amino)-N-(phenyloxyphenyl)acetamide structural motif representing a framework for selective SIRT2 inhibition.

  • Authors : Kaya SG; SIRTeam Group, Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Gazi University, Ankara, Türkiye.; Eren G

Subjects: Sirtuin 2*/Sirtuin 2*/Sirtuin 2*/antagonists & inhibitors ; Sirtuin 2*/Sirtuin 2*/Sirtuin 2*/chemistry ; Sirtuin 2*/Sirtuin 2*/Sirtuin 2*/metabolism

  • Source: Drug development research [Drug Dev Res] 2024 Jun; Vol. 85 (4), pp. e22224.Publisher: Wiley-Liss Country of Publication: United States NLM ID: 8204468 Publication Model: Print Cited Medium: Internet ISSN: 1098-2299

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Academic Journal

Dual-Mode Fluorescent/Intelligent Lateral Flow Immunoassay Based on Machine Learning Algorithm for Ultrasensitive Analysis of Chloroacetamide Herbicides.

  • Authors : Zha Y; State Key Laboratory for Diagnosis and Treatment of Severe Zoonotic Infectious Diseases, Key Laboratory for Zoonosis Research of the Ministry of Education, Institute of Zoonosis, and College of Veterinary Medicine, Jilin University, Changchun 130062, China.; School of Biomedical Engineering, Shenzhen Campus of Sun Yat-Sen University, Shenzhen 518107, China.

Subjects: Herbicides*/Herbicides*/Herbicides*/analysis ; Acetamides*/Acetamides*/Acetamides*/analysis ; Acetamides*/Acetamides*/Acetamides*/chemistry

  • Source: Analytical chemistry [Anal Chem] 2024 Jul 23; Vol. 96 (29), pp. 12197-12204. Date of Electronic Publication: 2024 Jul 11.Publisher: American Chemical Society Country of Publication: United States NLM ID: 0370536 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Design, synthesis, and biological evaluation of chalcone acetamide derivatives against triple negative breast cancer.

  • Authors : Kumar P; Natural Products and Medicinal Chemistry Division, CSIR - Indian Institute of Integrative Medicine, Jammu 180001, India; Academy of Scientific and Innovative Research (AcSIR), Ghaziabad 201002, India.

Subjects: Triple Negative Breast Neoplasms*/Triple Negative Breast Neoplasms*/Triple Negative Breast Neoplasms*/drug therapy ; Triple Negative Breast Neoplasms*/Triple Negative Breast Neoplasms*/Triple Negative Breast Neoplasms*/pathology ; Triple Negative Breast Neoplasms*/Triple Negative Breast Neoplasms*/Triple Negative Breast Neoplasms*/metabolism

  • Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2024 Jul 15; Vol. 107, pp. 129795. Date of Electronic Publication: 2024 May 13.Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Discovery of Novel 2-Oxoacetamide Derivatives as B3GAT3 Inhibitors for the Treatment of Hepatocellular Carcinoma.

  • Authors : Yin H; School of Science, China Pharmaceutical University, Nanjing 211198, China.; Zhang M

Subjects: Carcinoma, Hepatocellular*/Carcinoma, Hepatocellular*/Carcinoma, Hepatocellular*/drug therapy ; Carcinoma, Hepatocellular*/Carcinoma, Hepatocellular*/Carcinoma, Hepatocellular*/pathology ; Liver Neoplasms*/Liver Neoplasms*/Liver Neoplasms*/drug therapy

  • Source: Journal of medicinal chemistry [J Med Chem] 2024 Jul 11; Vol. 67 (13), pp. 10743-10773. Date of Electronic Publication: 2024 Jun 25.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Improved Radiosynthesis and Automation of [ 11 C]2-(2,6-Difluoro-4-((2-(N-methylphenylsulfonamido)ethyl)thio)phenoxy)acetamide ([ 11 C]K2) for Positron Emission Tomography of the Glutamate α-Amino-3-hydroxy-5-methyl-4-isoxazole Propionic Acid (AMPA) Receptor.

  • Authors : Witek JA; Department of Radiology, University of Michigan Medical School, Ann Arbor, Michigan, USA.; Horikawa M

Subjects: Positron-Emission Tomography*/Positron-Emission Tomography*/Positron-Emission Tomography*/methods ; Radiopharmaceuticals*/Radiopharmaceuticals*/Radiopharmaceuticals*/chemical synthesis ; Radiopharmaceuticals*/Radiopharmaceuticals*/Radiopharmaceuticals*/chemistry

  • Source: Journal of labelled compounds & radiopharmaceuticals [J Labelled Comp Radiopharm] 2024 Jul; Vol. 67 (9), pp. 324-329. Date of Electronic Publication: 2024 Jun 06.Publisher: Wiley Country of Publication: England NLM ID: 7610510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1099-1344

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Academic Journal

A real-world analysis of safety profile of selexipag by using FDA adverse Event Reporting System (FAERS).

  • Authors : Zhao J; Department of Pharmacy, Tongling People's Hospital, Tongling, Anhui Province, China.; Wang M

Subjects: Adverse Drug Reaction Reporting Systems*/Adverse Drug Reaction Reporting Systems*/Adverse Drug Reaction Reporting Systems*/statistics & numerical data ; United States Food and Drug Administration* ; Pyrazines*/Pyrazines*/Pyrazines*/adverse effects

  • Source: Expert opinion on drug safety [Expert Opin Drug Saf] 2024 Jul; Vol. 23 (7), pp. 937-948. Date of Electronic Publication: 2023 Dec 05.Publisher: Taylor & Francis Country of Publication: England NLM ID: 101163027 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Discovery of N-Substituted Acetamide Derivatives as Promising P2Y 14 R Antagonists Using Molecular Hybridization Based on Crystallographic Overlay.

  • Authors : Liu W; Henan Provincial Key Laboratory of Pediatric Hematology, Children's Hospital Affiliated to Zhengzhou University, Zhengzhou University, Zhengzhou 450018, China.; School of Pharmaceutical Science, Zhengzhou University, Zhengzhou 450001, China.

Subjects: Acetamides*/Acetamides*/Acetamides*/pharmacology ; Acetamides*/Acetamides*/Acetamides*/chemistry ; Acetamides*/Acetamides*/Acetamides*/chemical synthesis

  • Source: Journal of medicinal chemistry [J Med Chem] 2024 Jun 27; Vol. 67 (12), pp. 10233-10247. Date of Electronic Publication: 2024 Jun 14.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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  • 1-10 of  25,932 results for ""Acetamides""