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Academic Journal

Design, synthesis and biological evaluation of novel 6-phenyl-1,3a,4,10b-tetrahydro-2H-benzo[c]thiazolo[4,5-e]azepin-2-one derivatives as potential BRD4 inhibitors.

  • Authors : Li Q; Center of Drug Discovery, State Key Laboratory of Natural Medicine, China Pharmaceutical University, Nanjing 210009, PR China.; Li J

Subjects: Benzazepines/Benzazepines/Benzazepines/*pharmacology ; Cell Cycle Proteins/Cell Cycle Proteins/Cell Cycle Proteins/*antagonists & inhibitors ; Thiazoles/Thiazoles/Thiazoles/*pharmacology

  • Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2020 Aug 01; Vol. 28 (15), pp. 115601. Date of Electronic Publication: 2020 Jun 20.Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

The NPR1-WRKY46-WRKY6 signaling cascade mediates probenazole/salicylic acid-elicited leaf senescence in Arabidopsis thaliana.

  • Authors : Zhang D; State Key Laboratory of Genetic Engineering and Fudan Center for Genetic Diversity and Designing Agriculture, Institute of Plant Biology, School of Life Sciences, Fudan University, Shanghai, 200438, China.; Zhu Z

Subjects: Arabidopsis/Arabidopsis/Arabidopsis/*metabolism ; Arabidopsis/Arabidopsis/Arabidopsis/*physiology ; Arabidopsis Proteins/Arabidopsis Proteins/Arabidopsis Proteins/*metabolism

  • Source: Journal of integrative plant biology [J Integr Plant Biol] 2021 May; Vol. 63 (5), pp. 924-936. Date of Electronic Publication: 2021 Mar 08.Publisher: Wiley-Blackwell Pub Country of Publication: China (Republic : 1949- ) NLM ID: 101250502 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Differential Phosphorylation of the Transcription Factor WRKY33 by the Protein Kinases CPK5/CPK6 and MPK3/MPK6 Cooperatively Regulates Camalexin Biosynthesis in Arabidopsis.

  • Authors : Zhou J; Shanghai Key Laboratory of Plant Molecular Sciences, College of Life Sciences, Shanghai Normal University, Shanghai 200234, China.; Shanghai Key Laboratory of Bio-Energy Crops, School of Life Sciences, Shanghai University, Shanghai 200444, China.

Subjects: Biosynthetic Pathways*; Arabidopsis/Arabidopsis/Arabidopsis/*metabolism ; Arabidopsis Proteins/Arabidopsis Proteins/Arabidopsis Proteins/*metabolism Botrytis cinerea

  • Source: The Plant cell [Plant Cell] 2020 Aug; Vol. 32 (8), pp. 2621-2638. Date of Electronic Publication: 2020 May 21.Publisher: Oxford University Press Country of Publication: England NLM ID: 9208688 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

C-Myc inhibition sensitizes pre-B ALL cells to the anti-tumor effect of vincristine by altering apoptosis and autophagy: Proposing a probable mechanism of action for 10058-F4.

  • Authors : Sheikh-Zeineddini N; Department of Hematology and Blood Banking, School of Allied Medical Sciences, Shahid Beheshti University of Medical Sciences, Tehran, Iran.; Safaroghli-Azar A

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; DNA-Binding Proteins/DNA-Binding Proteins/DNA-Binding Proteins/*antagonists & inhibitors ; Precursor B-Cell Lymphoblastic Leukemia-Lymphoma/Precursor B-Cell Lymphoblastic Leukemia-Lymphoma/Precursor B-Cell Lymphoblastic Leukemia-Lymphoma/*drug therapy

  • Source: European journal of pharmacology [Eur J Pharmacol] 2020 Mar 05; Vol. 870, pp. 172821. Date of Electronic Publication: 2019 Nov 23.Publisher: Elsevier Science Country of Publication: Netherlands NLM ID: 1254354 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

New inhibitor targeting human transcription factor HSF1: effects on the heat shock response and tumor cell survival.

  • Authors : Vilaboa N; Hospital Universitario La Paz-IdiPAZ, 28046 Madrid, Spain.; CIBER de Bioingenieria, Biomateriales y Nanomedicina, CIBER-BBN, Madrid, Spain.

Subjects: Gene Expression Regulation, Neoplastic*; Acrylamides/Acrylamides/Acrylamides/*pharmacology ; Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology

  • Source: Nucleic acids research [Nucleic Acids Res] 2017 Jun 02; Vol. 45 (10), pp. 5797-5817.Publisher: Oxford University Press Country of Publication: England NLM ID: 0411011 Publication Model: Print Cited Medium: Internet ISSN:

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Academic Journal

ZY0511, a novel, potent and selective LSD1 inhibitor, exhibits anticancer activity against solid tumors via the DDIT4/mTOR pathway.

  • Authors : Li Y; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, West China Medical School, and Collaborative Innovation Center for Biotherapy, Sichuan University, Chengdu, 610041, China.; Tao L

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Enzyme Inhibitors/Enzyme Inhibitors/Enzyme Inhibitors/*pharmacology ; Histone Demethylases/Histone Demethylases/Histone Demethylases/*antagonists & inhibitors

  • Source: Cancer letters [Cancer Lett] 2019 Jul 10; Vol. 454, pp. 179-190. Date of Electronic Publication: 2019 Apr 10.Publisher: Elsevier Science Ireland Country of Publication: Ireland NLM ID: 7600053 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

In vitro-binding of the natural siderophore enantiomers pyochelin and enantiopyochelin to their AraC-type regulators PchR in Pseudomonas.

  • Authors : Lin PC; Département de Microbiologie Fondamentale, Université de Lausanne, Bâtiment Biophore, Quartier UNIL-Sorge, 1015, Lausanne, Switzerland.; Youard ZA

Subjects: Gene Expression Regulation, Bacterial*; Bacterial Proteins/Bacterial Proteins/Bacterial Proteins/*metabolism ; DNA-Binding Proteins/DNA-Binding Proteins/DNA-Binding Proteins/*metabolism

  • Source: Biometals : an international journal on the role of metal ions in biology, biochemistry, and medicine [Biometals] 2013 Dec; Vol. 26 (6), pp. 1067-73. Date of Electronic Publication: Publisher: Kluwer Academic Publishers Country of Publication: Netherlands NLM ID: 9208478 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Amino acid-derived 1,2-benzisothiazolinone derivatives as novel small-molecule antifungal inhibitors: identification of potential genetic targets.

Subjects: Amino Acids/Amino Acids/Amino Acids/*pharmacology ; Antifungal Agents/Antifungal Agents/Antifungal Agents/*pharmacology ; Fungal Proteins/Fungal Proteins/Fungal Proteins/*genetics

  • Source: Antimicrobial agents and chemotherapy [Antimicrob Agents Chemother] 2012 Sep; Vol. 56 (9), pp. 4630-9. Date of Electronic Publication: 2012 Jun 11.Publisher: American Society for Microbiology Country of Publication: United States NLM ID: 0315061 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

[Treatment with a tyrosine-kinase inhibitor of for c-KIT mutation and AML1-ETO double positive refractory acute myeloid leukemia].

  • Authors : Ueyama J; Tottori University, Division of Pediatrics and Perinatology.; Kure A

Subjects: Core Binding Factor Alpha 2 Subunit* ; Mutation* ; Proto-Oncogene Proteins*

  • Source: [Rinsho ketsueki] The Japanese journal of clinical hematology [Rinsho Ketsueki] 2012 Apr; Vol. 53 (4), pp. 460-4.Publisher: Japan Society Of Clinical Hematology Country of Publication: Japan NLM ID: 2984782R Publication Model: Print Cited Medium: Print ISSN:

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Academic Journal

Novel selective small molecule agonists for peroxisome proliferator-activated receptor delta (PPARdelta)--synthesis and biological activity.

  • Authors : Sznaidman ML; GlaxoSmithKline, Five Moore Drive, Research Triangle Park, NC 27709-3398, USA.; Haffner CD

Subjects: Receptors, Cytoplasmic and Nuclear/Receptors, Cytoplasmic and Nuclear/Receptors, Cytoplasmic and Nuclear/*agonists ; Thiazoles/Thiazoles/Thiazoles/*chemical synthesis ; Transcription Factors/Transcription Factors/Transcription Factors/*agonists

  • Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2003 May 05; Vol. 13 (9), pp. 1517-21.Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print Cited Medium: Print ISSN: 0960-894X

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  • 1-10 of  712 results for ""THIAZOLES""