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Joint toxic mechanism of clothianidin and prochloraz in the earthworm (Eisenia fetida).

• Authors : Liu X; State Key Laboratory for Managing Biotic and Chemical Threats to the Quality and Safety of Agro-products, Institute of Agro-product Safety and Nutrition, Zhejiang Academy of Agricultural Sciences, Hangzhou, 310021, Zhejiang, China.; Jia F

Subjects: Oligochaeta*/Oligochaeta*/Oligochaeta*/drug effects ; Neonicotinoids*/Neonicotinoids*/Neonicotinoids*/toxicity ; Thiazoles*/Thiazoles*/Thiazoles*/toxicity

• Source: Chemosphere [Chemosphere] 2024 Jul; Vol. 359, pp. 142250. Date of Electronic Publication: 2024 May 04.Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 0320657 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Development, synthesis and biological evaluation of imidazole [2,1-b] thiazole derivatives containing an indole ring for their potential anti-inflammatory properties.

• Authors : Jiang YC; Department of Pharmacy, Affiliated Hospital of Putian University, Putian, China.; Lin HF

Subjects: Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/pharmacology ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/chemical synthesis ; Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/Anti-Inflammatory Agents*/chemistry

• Source: Pakistan journal of pharmaceutical sciences [Pak J Pharm Sci] 2024 May; Vol. 37 (3), pp. 541-551.Publisher: Faculty of Pharmacy, University of Karachi Country of Publication: Pakistan NLM ID: 9426356 Publication Model: Print Cited Medium: Internet

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PERIOCULAR HIGH RISK BCCS AFTER ADDITIONAL/PARALLEL INTAKE OF TORASEMIDE, MOXONIDINE AND MIRABEGRON: IMPORTANT LINKS TO SKIN CANCER RELATED (PHOTO-) NITROSOGENESIS IN THE CONTEXT OF PHARMACO-ONCOGENESIS.

• Authors : Tchernev G; 1Onkoderma - Clinic for Dermatology, Venereology and Dermatologic Surgery, Sofia; 2Department of Dermatology and Venereology, Medical Institute of Ministry of Interior, Sofia, Bulgaria.

Subjects: Skin Neoplasms*/Skin Neoplasms*/Skin Neoplasms*/chemically induced ; Carcinoma, Basal Cell*/Carcinoma, Basal Cell*/Carcinoma, Basal Cell*/chemically induced ; Nitrosamines*/Nitrosamines*/Nitrosamines*/toxicity

• Source: Georgian medical news [Georgian Med News] 2024 Feb (347), pp. 70-76.Publisher: Assot︠s︡iat︠s︡ii︠a︡ delovoĭ pressy Gruzii Country of Publication: Georgia (Republic) NLM ID: 101218222 Publication Model: Print

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Design, synthesis and biological evaluation of 2,3-dihydroimidazo[2,1-b]thiazoles as dual EGFR and IGF1R inhibitors.

• Authors : Gadekar PK; Department of Medicinal Chemistry, Piramal Enterprises Limited, Goregaon (East), Mumbai 63, India; Center for Organic and Medicinal Chemistry, School of Advanced Sciences, VIT University, Vellore 632014, Tamil Nadu, India

Subjects: Drug Design*; Imidazoles/Imidazoles/Imidazoles/*chemistry ; Protein Kinase Inhibitors/Protein Kinase Inhibitors/Protein Kinase Inhibitors/*chemical synthesis

• Source: Bioorganic chemistry [Bioorg Chem] 2021 Oct; Vol. 115, pp. 105151. Date of Electronic Publication: 2021 Jul 07.Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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The architecture of hydrogen and sulfur σ-hole interactions explain differences in the inhibitory potency of C-β-d-glucopyranosyl thiazoles, imidazoles and an N-β-d glucopyranosyl tetrazole for human liver glycogen phosphorylase and offer new insights to structure-based design.

• Authors : Kyriakis E; Department of Biochemistry and Biotechnology, University of Thessaly, Biopolis, 41500 Larissa, Greece.; Karra AG

Subjects: Drug Design*; Enzyme Inhibitors/Enzyme Inhibitors/Enzyme Inhibitors/*pharmacology ; Glycogen Phosphorylase, Liver Form/Glycogen Phosphorylase, Liver Form/Glycogen Phosphorylase, Liver Form/*antagonists & inhibitors

• Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2020 Jan 01; Vol. 28 (1), pp. 115196. Date of Electronic Publication: 2019 Nov 14.Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Applied Science & Technology Full Text (H.W. Wilson)

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Nanomolar potency of imidazo[2,1-b]thiazole analogs as indoleamine 2,3-dioxygenase inhibitors.

• Authors : Ewida MA; Department of Pharmaceutical Chemistry, Faculty of Pharmaceutical Sciences & Pharmaceutical Industries, Future University in Egypt, Cairo, Egypt.; Ewida HA

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Imidazoles/Imidazoles/Imidazoles/*pharmacology ; Indoleamine-Pyrrole 2,3,-Dioxygenase/Indoleamine-Pyrrole 2,3,-Dioxygenase/Indoleamine-Pyrrole 2,3,-Dioxygenase/*antagonists & inhibitors

• Source: Archiv der Pharmazie [Arch Pharm (Weinheim)] 2021 Nov; Vol. 354 (11), pp. e2100202. Date of Electronic Publication: 2021 Jul 27.Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print-Electronic Cited Medium: Internet

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Novel imidazo[2,1-b]thiazole-based anticancer agents as potential focal adhesion kinase inhibitors: Synthesis, in silico and in vitro evaluation.

• Authors : Başoğlu F; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Istanbul University, Istanbul, Turkey.; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, European University of Lefke, Northern Cyprus, Turkey.

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*chemical synthesis ; Focal Adhesion Protein-Tyrosine Kinases/Focal Adhesion Protein-Tyrosine Kinases/Focal Adhesion Protein-Tyrosine Kinases/*antagonists & inhibitors ; Imidazoles/Imidazoles/Imidazoles/*chemistry

• Source: Chemical biology & drug design [Chem Biol Drug Des] 2021 Aug; Vol. 98 (2), pp. 270-282. Date of Electronic Publication: 2021 Jun 12.Publisher: Wiley-Blackwell Country of Publication: England NLM ID: 101262549 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Harmine-inspired design and synthesis of benzo[d]imidazo[2,1-b]thiazole derivatives bearing 1,3,4-oxadiazole moiety as potential tumor suppressors.

• Authors : Zhao T; Key Laboratory of Structure-Based Drug Design and Discovery, Ministry of Education, Shenyang Pharmaceutical University, Shenyang 110016, China.; Yang Y

Subjects: Drug Design*; Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Harmine/Harmine/Harmine/*pharmacology

• Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2021 Sep 15; Vol. 46, pp. 116367. Date of Electronic Publication: 2021 Aug 13.Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Discovery of New Imidazo[2,1- b ]thiazole Derivatives as Potent Pan-RAF Inhibitors with Promising In Vitro and In Vivo Anti-melanoma Activity.

• Authors : Abdel-Maksoud MS; Medicinal & Pharmaceutical Chemistry Department, Pharmaceutical and Drug Industries Research Division, National Research Centre (NRC), Dokki, Giza 12622, Egypt.; El-Gamal MI

Subjects: Imidazoles/Imidazoles/Imidazoles/*chemistry ; Protein Kinase Inhibitors/Protein Kinase Inhibitors/Protein Kinase Inhibitors/*chemistry ; Proto-Oncogene Proteins B-raf/Proto-Oncogene Proteins B-raf/Proto-Oncogene Proteins B-raf/*antagonists & inhibitors

• Source: Journal of medicinal chemistry [J Med Chem] 2021 May 27; Vol. 64 (10), pp. 6877-6901. Date of Electronic Publication: 2021 May 17.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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