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Solid-phase synthesis of curcumin mimics and their anticancer activity against human pancreatic, prostate, and colorectal cancer cell lines.

• Authors : Romanucci V; Department of Chemical Sciences, University of Napoli Federico II, Via Cintia 4, 80126 Napoli, Italy.; Giordano M

Subjects: Solid-Phase Synthesis Techniques*; Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Curcumin/Curcumin/Curcumin/*pharmacology

• Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2021 Jul 15; Vol. 42, pp. 116249. Date of Electronic Publication: 2021 Jun 05.Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Synthesis and SAR Analysis of Lipovelutibols B and D and Their Lipid Analogues.

• Authors : Cameron AJ; School of Chemical Sciences , University of Auckland , 23 Symonds Street , Auckland , 1010 , New Zealand.; School of Biological Sciences , University of Auckland , 3 Symonds Street , Auckland , 1010 , New Zealand.

Subjects: Antineoplastic Agents* ; Solid-Phase Synthesis Techniques*; Lipids

• Source: The Journal of organic chemistry [J Org Chem] 2020 Feb 07; Vol. 85 (3), pp. 1401-1406. Date of Electronic Publication: 2019 Dec 06.Publisher: American Chemical Society Country of Publication: United States NLM ID: 2985193R Publication Model: Print-Electronic Cited Medium: Internet

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Parallel Solid-Phase Synthesis using a New Diethylsilylacetylenic Linker and Leading to Mestranol Derivatives with Potent Antiproliferative Activities on Multiple Cancer Cell Lines.

• Authors : Dutour R; Laboratory of Medicinal Chemistry, Endocrinology and Nephrology Unit, CHU de Quebec-Research Center (CHUL-T4), Quebec, QC, Canada.; Department of Molecular Medicine, Faculty of Medicine, Université Laval, Québec, QC, Canada.

Subjects: Solid-Phase Synthesis Techniques*; Acetylene/Acetylene/Acetylene/*pharmacology ; Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology

• Source: Anti-cancer agents in medicinal chemistry [Anticancer Agents Med Chem] 2018; Vol. 18 (10), pp. 1469-1481.Publisher: Bentham Science Publishers Country of Publication: Netherlands NLM ID: 101265649 Publication Model: Print Cited Medium: Internet ISSN:

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Facial Solid-Phase Synthesis of Well-Defined Zwitterionic Amphiphiles for Enhanced Anticancer Drug Delivery.

• Authors : Wang L; Ji X; Guo D

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*administration & dosage ; Doxorubicin/Doxorubicin/Doxorubicin/*administration & dosage ; Nanoparticle Drug Delivery System/Nanoparticle Drug Delivery System/Nanoparticle Drug Delivery System/*chemical synthesis

• Source: Molecular pharmaceutics [Mol Pharm] 2021 Jun 07; Vol. 18 (6), pp. 2349-2359. Date of Electronic Publication: 2021 May 13.Publisher: American Chemical Society Country of Publication: United States NLM ID: 101197791 Publication Model: Print-Electronic Cited Medium: Internet

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Bioconjugates of Co(III) complexes with Schiff base ligands and cell penetrating peptides: Solid phase synthesis, characterization and antiproliferative activity.

• Authors : Śmiłowicz D; Inorganic Chemistry I - Bioinorganic Chemistry, Ruhr-University Bochum, Universitätsstraße 150, 44801 Bochum, Germany.; Metzler-Nolte N

Subjects: Cell Proliferation*; Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*pharmacology ; Cell-Penetrating Peptides/Cell-Penetrating Peptides/Cell-Penetrating Peptides/*chemistry

• Source: Journal of inorganic biochemistry [J Inorg Biochem] 2020 May; Vol. 206, pp. 111041. Date of Electronic Publication: 2020 Feb 20.Publisher: Elsevier Country of Publication: United States NLM ID: 7905788 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Preparation of Enzyme-Activated Thapsigargin Prodrugs by Solid-Phase Synthesis.

• Authors : Zimmermann T; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Jagtvej 162, DK-2100 Copenhagen, Denmark. .; Christensen SB

Subjects: Antineoplastic Agents/Antineoplastic Agents/Antineoplastic Agents/*chemical synthesis ; Prodrugs/Prodrugs/Prodrugs/*chemical synthesis ; Solid-Phase Synthesis Techniques/Solid-Phase Synthesis Techniques/Solid-Phase Synthesis Techniques/*methods

• Source: Molecules (Basel, Switzerland) [Molecules] 2018 Jun 15; Vol. 23 (6). Date of Electronic Publication: 2018 Jun 15.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Solid-phase synthesis and pharmacological evaluation of novel nucleoside-tethered dinuclear platinum(II) complexes.

• Authors : D'Errico S; Dipartimento di Chimica delle Sostanze Naturali, Università degli Studi di Napoli Federico II, Via D. Montesano 49, 80131 Napoli, Italy. ; Oliviero G

Subjects: Solid-Phase Synthesis Techniques*; Antimetabolites, Antineoplastic/Antimetabolites, Antineoplastic/Antimetabolites, Antineoplastic/*chemical synthesis ; Antimetabolites, Antineoplastic/Antimetabolites, Antineoplastic/Antimetabolites, Antineoplastic/*pharmacology

• Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2011 Oct 01; Vol. 21 (19), pp. 5835-8. Date of Electronic Publication: 2011 Aug 03.Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Solid-Phase Synthesis of Cereblon-Recruiting Selective Histone Deacetylase 6 Degraders (HDAC6 PROTACs) with Antileukemic Activity.

• Authors : Sinatra L; Institute for Drug Discovery, Medical Faculty, Leipzig University, Brüderstrasse 34, 04103 Leipzig, Germany.; Yang J

Subjects: Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/pharmacology; Histone Deacetylase 6 ; Proteolysis Targeting Chimera

• Source: Journal of medicinal chemistry [J Med Chem] 2022 Dec 22; Vol. 65 (24), pp. 16860-16878. Date of Electronic Publication: 2022 Dec 06.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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Novel Approaches for the Solid-Phase Synthesis of Dihydroquinazoline-2(1 H )-One Derivatives and Biological Evaluation as Potential Anticancer Agents.

• Authors : Wang Q; Department of Chemistry, Shantou University Medical College, 22 Xinling Road, Shantou 515041, China.; National Cancer Center/National Clinical Research Center for Cancer/Cancer Hospital & Shenzhen Hospital, Chinese Academy of Medical Sciences and Peking Union Medical College, Shenzhen 518116, China.

Subjects: Ovarian Neoplasms* ; Antineoplastic Agents*/Antineoplastic Agents*/Antineoplastic Agents*/chemistry; Female

• Source: Molecules (Basel, Switzerland) [Molecules] 2022 Dec 05; Vol. 27 (23). Date of Electronic Publication: 2022 Dec 05.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Agricola

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