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Academic Journal

Chemical evidence for the difference between albumins from microsomes and serum and a possible precursor-product relationship.

Subjects: Albumins*/Albumins*/Albumins*/analysis ; Albumins*/Albumins*/Albumins*/isolation & purification ; Serum Albumin*/Serum Albumin*/Serum Albumin*/analysis

  • Source: Biochemical and biophysical research communications [Biochem Biophys Res Commun] 1974 Nov 27; Vol. 61 (2), pp. 494-501.Publisher: Elsevier Country of Publication: United States NLM ID: 0372516 Publication Model: Print Cited Medium: Print

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Academic Journal

Effects of species of origin and mode of induction of microsomes on carbamazepine-induced cell toxicity.

  • Authors : Elzagallaai AA; Department of Paediatrics, Schulich School of Medicine and Dentistry, University of Western Ontario, London, Ontario, Canada; Department of Physiology and Pharmacology, Schulich School of Medicine and Dentistry, University of Western Ontario, London, Ontario, Canada

Subjects: Carbamazepine*/Carbamazepine*/Carbamazepine*/toxicity ; Microsomes, Liver*/Microsomes, Liver*/Microsomes, Liver*/drug effects ; Microsomes, Liver*/Microsomes, Liver*/Microsomes, Liver*/metabolism

  • Source: Journal of pharmacological and toxicological methods [J Pharmacol Toxicol Methods] 2024 Jul-Aug; Vol. 128, pp. 107536. Date of Electronic Publication: 2024 Jul 05.Publisher: Elsevier Country of Publication: United States NLM ID: 9206091 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

In vitro characterization of protonitazene metabolites, using human liver microsomes, and first application to two urines collected from death cases.

  • Authors : Ameline A; Institut de Médecine Légale, 11 rue Humann, 67085 Strasbourg, France. Electronic address: .; Gheddar L

Subjects: Microsomes, Liver*/Microsomes, Liver*/Microsomes, Liver*/metabolism ; Microsomes, Liver*/Microsomes, Liver*/Microsomes, Liver*/chemistry ; Benzimidazoles*/Benzimidazoles*/Benzimidazoles*/metabolism

  • Source: Clinica chimica acta; international journal of clinical chemistry [Clin Chim Acta] 2024 Jul 15; Vol. 561, pp. 119764. Date of Electronic Publication: 2024 Jun 04.Publisher: Elsevier Country of Publication: Netherlands NLM ID: 1302422 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Effects of the antitumor drugs adagrasib and asciminib on apixaban metabolism in vitro and in vivo.

  • Authors : Shen Y; Department of Pharmacy, The First Affiliated Hospital of Wenzhou Medical University, Wenzhou, Zhejiang, China; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.

Subjects: Pyrazoles*/Pyrazoles*/Pyrazoles*/pharmacology ; Pyrazoles*/Pyrazoles*/Pyrazoles*/metabolism ; Pyridones*/Pyridones*/Pyridones*/pharmacology

  • Source: Chemico-biological interactions [Chem Biol Interact] 2024 Aug 25; Vol. 399, pp. 111146. Date of Electronic Publication: 2024 Jul 14.Publisher: Elsevier Country of Publication: Ireland NLM ID: 0227276 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Inhibitory effect of imperatorin on dabrafenib metabolism in vitro and in vivo.

  • Authors : Xia H; Department of Pharmacy, The First Affiliated Hospital of Wenzhou Medical University, Wenzhou, Zhejiang, China.; Wu H

Subjects: Oximes*/Oximes*/Oximes*/pharmacology ; Imidazoles*/Imidazoles*/Imidazoles*/pharmacology ; Imidazoles*/Imidazoles*/Imidazoles*/metabolism

  • Source: Chemico-biological interactions [Chem Biol Interact] 2024 Aug 25; Vol. 399, pp. 111131. Date of Electronic Publication: 2024 Jul 02.Publisher: Elsevier Country of Publication: Ireland NLM ID: 0227276 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Ultra-fast UPLC-MS/MS approach for estimating X-376 in human liver microsomes: Evaluation of metabolic stability via in silico software and in vitro analysis.

  • Authors : Attwa MW; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia.. Electronic address: .; Abdelhameed AS

Subjects: Tandem Mass Spectrometry*/Tandem Mass Spectrometry*/Tandem Mass Spectrometry*/methods ; Microsomes, Liver*/Microsomes, Liver*/Microsomes, Liver*/metabolism ; Software*

  • Source: Journal of pharmacological and toxicological methods [J Pharmacol Toxicol Methods] 2024 Jul-Aug; Vol. 128, pp. 107540. Date of Electronic Publication: 2024 Jul 10.Publisher: Elsevier Country of Publication: United States NLM ID: 9206091 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Comparison of Commonly Used and New Methods to Determine Small Molecule Non-Specific Binding to Human Liver Microsomes.

  • Authors : Wang T; Department of Drug Metabolism and Pharmacokinetics, Boehringer Ingelheim Pharmaceuticals Inc., 900 Ridgebury Rd., Ridgefield, CT 06877, USA. Electronic address: .; Whitcher-Johnstone A

Subjects: Microsomes, Liver*/Microsomes, Liver*/Microsomes, Liver*/metabolism ; Ultrafiltration*/Ultrafiltration*/Ultrafiltration*/methods; Humans

  • Source: Journal of pharmaceutical sciences [J Pharm Sci] 2024 Jul; Vol. 113 (7), pp. 1987-1995. Date of Electronic Publication: 2024 Apr 12.Publisher: Elsevier Country of Publication: United States NLM ID: 2985195R Publication Model: Print-Electronic Cited Medium:

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Academic Journal

In vitro demonstration of antedrug mechanism of a pharmacokinetic booster to improve CYP3A4 substrates by CYP3A4-mediated metabolism inhibition.

  • Authors : Kataoka M; Faculty of Pharmaceutical Sciences, Setsunan University, 45-1 Nagaotoge-cho, Hirakata, Osaka, 573-0101, Japan. Electronic address: .; Takenaka S

Subjects: Cytochrome P-450 CYP3A*/Cytochrome P-450 CYP3A*/Cytochrome P-450 CYP3A*/metabolism ; Microsomes, Liver*/Microsomes, Liver*/Microsomes, Liver*/metabolism ; Midazolam*/Midazolam*/Midazolam*/metabolism

  • Source: Drug metabolism and pharmacokinetics [Drug Metab Pharmacokinet] 2024 Jun; Vol. 56, pp. 101005. Date of Electronic Publication: 2024 Mar 02.Publisher: Elsevier Country of Publication: England NLM ID: 101164773 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Inhibition of soluble epoxide hydrolase by natural isothiocyanates.

  • Authors : Elbarbry F; School of Pharmacy, Pacific University, 222 SE 8th Ave, Ste. 451, Hillsboro, OR, 97123, USA. Electronic address: .; Espiritu MJ

Subjects: Epoxide Hydrolases*/Epoxide Hydrolases*/Epoxide Hydrolases*/antagonists & inhibitors ; Epoxide Hydrolases*/Epoxide Hydrolases*/Epoxide Hydrolases*/metabolism ; Epoxide Hydrolases*/Epoxide Hydrolases*/Epoxide Hydrolases*/chemistry

  • Source: Biochemical and biophysical research communications [Biochem Biophys Res Commun] 2024 Sep 17; Vol. 725, pp. 150261. Date of Electronic Publication: 2024 Jun 12.Publisher: Elsevier Country of Publication: United States NLM ID: 0372516 Publication Model: Print-Electronic Cited Medium:

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Academic Journal

Metabolic transformation of cyclopiazonic acid in liver microsomes from different species based on UPLC-Q/TOF-MS.

  • Authors : Ye Y; School of Food Science and Technology, International Joint Laboratory on Food Safety, Synergetic Innovation Center of Food Safety and Quality Control, Jiangnan University, Wuxi, Jiangsu 214122, PR China.; Sun X

Subjects: Microsomes, Liver*/Microsomes, Liver*/Microsomes, Liver*/metabolism ; Indoles*/Indoles*/Indoles*/metabolism; Animals

  • Source: Journal of hazardous materials [J Hazard Mater] 2024 Sep 05; Vol. 476, pp. 134902. Date of Electronic Publication: 2024 Jun 13.Publisher: Elsevier Country of Publication: Netherlands NLM ID: 9422688 Publication Model: Print-Electronic Cited Medium:

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