Search Results

Filter
  • 1-10 of  135 results for ""NOOTROPIC agents""
Item request has been placed! ×
Item request cannot be made. ×
loading  Processing Request
Academic Journal

A new arylsulfanyl-benzo-2,1,3-thiadiazoles derivative produces an anti-amnesic effect in mice by modulating acetylcholinesterase activity.

  • Authors : da Costa Rodrigues K; Postgraduate Program in Biochemistry and Bioprospecting, Research Laboratory in Biochemical Pharmacology (LaFarBio), Research Group in Neurobiotechnology (GPN), Center of Chemical, Pharmaceutical and Food Sciences, Federal University of Pelotas (UFPel), CEP 96010- 900, Pelotas, RS, Brazil.; Leivas de Oliveira R

Subjects: Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*metabolism ; Amnesia/Amnesia/Amnesia/*drug therapy ; Cholinesterase Inhibitors/Cholinesterase Inhibitors/Cholinesterase Inhibitors/*therapeutic use

  • Source: Chemico-biological interactions [Chem Biol Interact] 2022 Jan 05; Vol. 351, pp. 109736. Date of Electronic Publication: 2021 Nov 03.Publisher: Elsevier Country of Publication: Ireland NLM ID: 0227276 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-7786

Record details

×
Academic Journal

Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate.

  • Authors : Zhou Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai 201203, People's Republic of China.; School of Pharmacy, University of Chinese Academy of Sciences, No. 19A Yuquan Road, Beijing 100049, People's Republic of China.

Subjects: Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*metabolism ; Cholinesterase Inhibitors/Cholinesterase Inhibitors/Cholinesterase Inhibitors/*therapeutic use ; Indans/Indans/Indans/*therapeutic use

  • Source: Journal of medicinal chemistry [J Med Chem] 2021 Feb 25; Vol. 64 (4), pp. 1844-1855. Date of Electronic Publication: 2021 Feb 11.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

Record details

×
Academic Journal

Usnic acid enantiomers restore cognitive deficits and neurochemical alterations induced by Aβ 1-42 in mice.

  • Authors : Cazarin CA; Pharmaceutical Sciences Postgraduate Program, Center of Health Sciences, Universidade do Vale do Itajaí, CEP 88302-202, Itajaí, Santa Catarina, Brazil. Electronic address: .; Dalmagro AP

Subjects: Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*drug effects ; Alzheimer Disease/Alzheimer Disease/Alzheimer Disease/*drug therapy ; Amyloid beta-Peptides/Amyloid beta-Peptides/Amyloid beta-Peptides/*pharmacology

  • Source: Behavioural brain research [Behav Brain Res] 2021 Jan 15; Vol. 397, pp. 112945. Date of Electronic Publication: 2020 Oct 03.Publisher: Elsevier/North-Holland Biomedical Press Country of Publication: Netherlands NLM ID: 8004872 Publication Model: Print-Electronic Cited Medium:

Record details

×
Academic Journal

Cholinesterase inhibitors as Alzheimer's therapeutics (Review).

  • Authors : Sharma K; Department of Chemistry, Faculty of Physical Sciences, Shree Guru Gobind Singh Tricentenary University, Gurugram, Haryana 122505, India.

Subjects: Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*metabolism ; Alzheimer Disease/Alzheimer Disease/Alzheimer Disease/*drug therapy ; Choline/Choline/Choline/*metabolism

  • Source: Molecular medicine reports [Mol Med Rep] 2019 Aug; Vol. 20 (2), pp. 1479-1487. Date of Electronic Publication: 2019 Jun 11.Publisher: D. A. Spandidos Country of Publication: Greece NLM ID: 101475259 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

Record details

×
Academic Journal

The acetylcholinesterase (AChE) inhibitor and anti-Alzheimer drug donepezil interacts with human erythrocytes.

  • Authors : Zambrano P; Facultad de Ciencias Químicas, Universidad de Concepción, Concepción, Chile.; Suwalsky M

Subjects: Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*drug effects ; Alzheimer Disease/Alzheimer Disease/Alzheimer Disease/*drug therapy ; Cholinesterase Inhibitors/Cholinesterase Inhibitors/Cholinesterase Inhibitors/*pharmacology

  • Source: Biochimica et biophysica acta. Biomembranes [Biochim Biophys Acta Biomembr] 2019 Jun 01; Vol. 1861 (6), pp. 1078-1085. Date of Electronic Publication: 2019 Mar 20.Publisher: Elsevier Country of Publication: Netherlands NLM ID: 101731713 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

Record details

×
Academic Journal

New semicarbazones as gorge-spanning ligands of acetylcholinesterase and potential new drugs against Alzheimer's disease: Synthesis, molecular modeling, NMR, and biological evaluation.

  • Authors : Ferreira Neto DC; a Medicinal Chemistry Group , Military Institute of Engineering , Praia Vermelha, Rio de Janeiro 22290-270 , Brazil.; b Department of Chemistry , Federal University of Roraima , Boa Vista, Roraima 69310-000 , Brazil.

Subjects: Molecular Dynamics Simulation*; Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*chemistry ; Nootropic Agents/Nootropic Agents/Nootropic Agents/*chemical synthesis

  • Source: Journal of biomolecular structure & dynamics [J Biomol Struct Dyn] 2018 Nov; Vol. 36 (15), pp. 4099-4113. Date of Electronic Publication: 2017 Dec 07.Publisher: Taylor & Francis Country of Publication: England NLM ID: 8404176 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

Record details

×
Academic Journal

Exploiting the Chalcone Scaffold to Develop Multifunctional Agents for Alzheimer's Disease.

  • Authors : Rampa A; Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, Via Belmeloro 6, 40126 Bologna, Italy. .; Bartolini M

Subjects: Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*chemistry ; Antioxidants/Antioxidants/Antioxidants/*chemical synthesis ; Butyrylcholinesterase/Butyrylcholinesterase/Butyrylcholinesterase/*chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2018 Jul 30; Vol. 23 (8). Date of Electronic Publication: 2018 Jul 30.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

Record details

×
Academic Journal

Characterization of the interactions between coumarin-derivatives and acetylcholinesterase: Examination by NMR and docking simulations.

  • Authors : Tanoli NU; Department of Metallurgy and Materials Engneering, Pakistan Institute of Engineering and Applied Sciences (PIEAS), Lehtrar Road, Nilore, Islamabad, 45650, Pakistan. .; Laboratory of Nuclear Magnetic Resonance, Federal University of São Carlos, Rodovia Washington Luiz, Km 235, São Carlos, SP, 13565-905, Brazil. .

Subjects: Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*chemistry ; Cholinesterase Inhibitors/Cholinesterase Inhibitors/Cholinesterase Inhibitors/*chemistry ; Coumarins/Coumarins/Coumarins/*chemistry

  • Source: Journal of molecular modeling [J Mol Model] 2018 Jul 14; Vol. 24 (8), pp. 207. Date of Electronic Publication: 2018 Jul 14.Publisher: Springer Country of Publication: Germany NLM ID: 9806569 Publication Model: Electronic Cited Medium: Internet ISSN: 0948-5023

Record details

×
Academic Journal

Synthesis and biological evaluation of ranitidine analogs as multiple-target-directed cognitive enhancers for the treatment of Alzheimer's disease.

  • Authors : Gao J; Drug Discovery and Biomedical Sciences, South Carolina College of Pharmacy, University of South Carolina, Columbia, SC 29208, USA; Department of Pharmacology and Toxicology, Augusta University, Health Sciences Campus, CB-3530, 1459 Laney Walker Blvd., Augusta, GA 30912, USA.

Subjects: Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*metabolism ; Cholinesterase Inhibitors/Cholinesterase Inhibitors/Cholinesterase Inhibitors/*chemistry ; Cholinesterase Inhibitors/Cholinesterase Inhibitors/Cholinesterase Inhibitors/*pharmacology

  • Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2016 Nov 15; Vol. 26 (22), pp. 5573-5579. Date of Electronic Publication: 2016 Oct 06.Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

Record details

×
Academic Journal

Amino acid content and acetylcholinesterase inhibition of Huperzia saururus infusion and decoction.

  • Authors : Vallejo MG; Department of Pharmacy, School of Chemical Sciences, National University of Córdoba, IMBIV-CONICET, Córdoba, Argentina.; Dimmer JA

Subjects: Huperzia*/Huperzia*/Huperzia*/chemistry; Acetylcholinesterase/Acetylcholinesterase/Acetylcholinesterase/*metabolism ; Arginine/Arginine/Arginine/*pharmacology

  • Source: Pharmaceutical biology [Pharm Biol] 2013 Oct; Vol. 51 (10), pp. 1341-5. Date of Electronic Publication: 2013 Jul 10.Publisher: Taylor & Francis Country of Publication: England NLM ID: 9812552 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

Record details

×
  • 1-10 of  135 results for ""NOOTROPIC agents""